List of Publications

154Site-Selective Functionalization of Cysteine Units in Peptides Through Meerwein Arylation Reactions Under Mild Conditions
D. R. Troeger, N. Diesendorf, R. Thurston, M. R. Heinrich, Synth. Catal, 2026, 368, e70594.
DOI: 10.1002/adsc.70594
153The FAU expired drug initiative (FAU EDI) – recovery of APIs from expired drugs to support research and teaching in Europe
L. E. F. Lochschmidt, E. Winter, M. Kuschow, A. Roggenhofer, M. R. Heinrich, Sustainable Chemistry and Pharmacy, 2026, 52, 102463.
DOI: 10.1016/j.scp.2026.102463
152Synthesis and Evaluation of Novel Sulfonamido-oxine (Sox)-Substituted Lysine Derivatives
M. Kuschow, J. Kuhn, L. Drees, L. Schuster, V. Osterloh, M. R. Heinrich, Synthesis, 2026.
DOI: 10.1055/a-2872-0385
151Total Synthesis of rac-Keramamine C Enabled by Intrinsic H-Bond-Induced Conformational Fixation of Amides
J. Ganzmann, R. Thurston, P. Riester, N. Hegmann, M. R. Heinrich, European Journal of Organic Chemistry, 2026, 29, e202501128.
DOI: 10.1002/ejoc.202501128
150In vitro transporter substrate properties of previously reported biomarkers for renal OAT1/OAT3-mediated drug-drug interactions
J. Picurová, A. Gessner, N. Bartels, S. Scheuerlein, O. Fischer, L. E. F. Lochschmidt, P. Wenisch, P. Stopfer, M. R. Heinrich, J. König, M. F. Fromm, Biochemical Pharmacology, 2025, 241, 117184.
DOI: 10.1016/j.bcp.2025.117184
1493,4,5-Trifluorophenyldiazonium a unique radical source for the visible light induced, catalyst-free arylation of tyrosine residues in peptides
M. Kuschow, D. Troeger, L.-S. Schuster, L. Bock, L. Z hnle, M. R. Heinrich, Chem. Eur. J., 2025, 31, 38.
DOI: 10.1002/chem.202501160
148Controlled Growth of Oligophenylene-Structures on Graphene for Facile Secondary functionalization
C. E. Halbig, F. Fels, S. Wei, R. Schusterbauer, I. Donskyi, M. R. Heinrich, S. Eigler, Angew. Chem. Int. Ed., 2025, 64, 25.
DOI: 10.1002/anie.202504482
147Enzymatically formed fatty acid hydroperoxides determined through GC-MS analysis of enantiomeric excess of hydroxy fatty acids after reduction and ibuprofen derivatization
L. Hotz, A. Zartmann, Luca J. Drees, M. K. Kuschow, M. R. Heinrich, H-G. Janssen, S. Hammann, Eur. J. Lipid Sci. Technol., 2025, 127, 2.
DOI: 10.1002/ejlt.202400065
146An untargeted metabolomics approach to evaluate enzymatically deconjugated steroids and intact steroid conjugates in urine as diagnostic biomarkers for adrenal tumors
N. Vogg, E. North, A. Gessner, F. Fels, M. R. Heinrich, M. Kroiss, M. Kurlbaum, M. Fassnacht, M. F. Fromm, Clin. Chem. Lab. Med., 2025, 63, 1004-1015.
DOI: 10.1515/cclm-2024-1337
145Dually labeled neurotensin NTS1R ligands for probing radiochemical and fluorescence-based binding assays
F. Ertl, S. Kopanchuk, N. C. Dijon, S. Veik ina, M.-J. Tahk, T. Laasfeld, F. Schettler, A. O. Gattor, H. H bner, N. Archipowa, J. K ckenberger, M. R. Heinrich, P. Gmeiner, R.-J. Kutta, N. D. Holliday, A. Rinken, M. Keller, J. Med. Chem., 2024, 67, 18.
DOI: 10.1021/acs.jmedchem.4c01470
144Identification of novel inhibitors of the transcriptional coactivator MRTF-A for HCC therapy
M. J. Franz, P. Wenisch, P. Wohlleben, V. Chubanov, T. Gudermann, S. Kyher inen, M. Vartiainen, M. R. Heinrich, S. Muehlich, Mol. Ther. Oncol., 2024, 32, 3, 200855.
DOI: 10.1016/j.omton.2024.200855
143New biomarkers for renal transporter-mediated drug-drug interactions: metabolomic effects of cimetidine, probenecid, verapamil, and rifampin in humans
A. Gessner, J. König, P. Wenisch, M. R. Heinrich, P. Stopfer, M. F. Fromm, F. M ller, Clin. Pharmacol. Ther., 2024,
DOI: 10.1002/cpt.3414
142Illuminating neuropeptide Y Y4 receptor binding: fluorescent cyclic peptides with subnanomolar binding affinity as novel molecular tools
J. Gleixner, S. Kopanchuk, L. Gr tz, M.-J. Tahk, T. Laasfeld, S. Veiksina, C. H ring, A. Gattor, L. Humphrys, C. M ller, N. Archipowa, J. K ckenberger, M. R. Heinrich, R.-J. Kutta, A. Rinken, M. Keller, ACS Pharmacol. Transl. Sci., 2024, 7, 4, 1142-1168.
DOI: 10.1021/acsptsci.4c00013
141Visible light-mediated catalyst-free radical arylations using arenediazonium salts
P. Wenisch, M. Kuschow, M. R. Heinrich, Arkivoc, 2024, 202312113(special issue in the honour of Prof. Samir Zard)
DOI: 10.24820/ark.5550190.p012.113
140Characterization of fluorescent dyes frequently used for bioimaging: photophysics and photocatalytical reactions with protein
N. Archipowa, L. Wittmann, J. K ckenberger, F. J. Ertl, J. Gleixner, M. Keller, M. R. Heinrich, R.-J. Kutta, J. Phys. Chem. B., 2023, 127, 44, 9532-9542.
DOI: 10.1021/acs.jpcb.3c04484
139Labor statt M llcontainer
M. R. Heinrich, Nachrichten aus der Chemie, October 2023, 71, 10, S.36-37.
DOI: 10.1002/nadc.20234138226
138A metabolomic analysis of sensitivity and specificity of 23 previously proposed biomarkers for renal transporter-mediated drug-drug interactions
A. Gessner, F. M ller, P. Wenisch, M. R. Heinrich, J. K nig, P. Stopfer, M. F. Fromm, Clin. Pharmacol. Ther., 2023, 114, 5.
DOI: 10.1002/cpt.3017
137Electrophotographic 3D printing of pharmaceutical films
S.-P. Kopp, V. Medvedev, K. Tangermann-Gerk, N. W ltinger, R. Rothfelder, F. Gra l, M. R. Heinrich, P. Januskaite, A. Goyanes, A. W. Basit, S. Roth, M. Schmidt, Addit. Manuf., 2023, 73, 103707.
DOI: 10.1016/j.addma.2023.103707
136Exploring structural determinants of bias among D4 subtype-selective dopamine receptor agonists
F. Graßl, L. Bock, A. H.-H. Gonzalez, M. Schiller, P. Gmeiner, J. K nig, M. F. Fromm, H. H bner, M. R. Heinrich, J. Med. Chem., 2023, 66, 14, 9710-9730.
DOI: 10.1021/acs.jmedchem.3c00537
135Tuning the Polarity of Antibiotic-Cy5 Conjugates Enables Highly Selective Labeling of Binding Sites
F. Graßl, M. B. Konrad, J. Kr ll, A. Pezerovic, L. Z hnle, A. Burkovski, M. R. Heinrich, Chem. Eur. J., 2023, 29, 45.
DOI: 10.1002/chem.202301208
134Identification and Quantification of Resveratrol and Its Derivatives in Franconian Wines by Comprehensive Liquid Chromatography Tandem Mass Spectrometry
L. Hoferer, V. Rodrigues Guimaraes Abreu, F. Gra l, O. Fischer, M. R. Heinrich, S. Gensberger-Reigl, ACS Food Sci. Technol., 2023, 3, 6, 1057-1067.
DOI: 10.1021/acsfoodscitech.3c00070
133Connecting Ruthenium Photocatalysis to 1,2-Dioxetane-Mediated Chemiluminescence: a Versatile Combination for Optical Detection and Read-Out
J. Köckenberger, R. Thurston, C. Sauer, J. Oppl, M. R. Heinrich, Angew. Chem. Int. Ed., 2023, 62, 31.
DOI: 10.1002/anie.202304474
132Cyanine- and Rhodamine-Derived Alkynes for the Selective Targeting of Cancerous Mitochondria via Radical Thiol-Yne Coupling in Live Cells
J. Köckenberger, I. Klemt, C. Sauer, A. Arkhypov, V. Reshetnikov, A. Mokhir, M. R. Heinrich, Chem. Eur. J., 2023, 29, 45.
DOI: 10.1002/chem.202301340
131Selectfluor-mediated chlorination and fluorination of arenes: late stage functionalization of APIs and its biological effects
S. Gradl, V. Zantop, P. Gmeiner, H. H bner, M. R. Heinrich, ChemMedChem, 2023, 18, 15.
DOI: 10.1002/cmdc.202300144
130Behaviour effects of APH199, a selective dopamine D4 receptor agonist, in animal models
D. Chestnykh, F. Gra l, C. Pfeifer, J. D lk, C. Ebner, M. Walters, S. von H rsten, J. Kornhuber, L. S. Kalinichenko, M. R. Heinrich, C. P. M ller, Psychopharmacology, 2023, 240, 1011-1031.
DOI: 10.1007/s00213-023-06347-1
129Visible-light mediated radical arylations using a fluorescein-derived diazonium salt: reactions proceeding via an intramolecular forth and back electron transfer
N. Diesendorf, P. Wenisch, J. Oppl, M. R. Heinrich, Org. Lett., 2023, 25, 1, 76-81.
DOI: 10.1021/acs.orglett.2c03877
128Synthesis, characterization and application of muscarinergic M3 receptor ligands linked to fluorescent dyes
J. Köckenberger, O. Fischer, A. Konopa, S. Bergwinkl, S. Mühlich, P. Gmeiner, R. J. Kutta, H. H bner, M. Keller, M. R. Heinrich , J. Med. Chem., 2022, 65, 24, 16494-16509.
DOI: 10.1021/acs.jmedchem.2c01376
127Analysis of hyperforin (St John s wort) action at TRPC6 channel leads to the development of new antidepressant drugs
Y. E. Hamdaoui, F. Zheng, N. Fritz, L. Ye, M. A. Tran, K. Schwickert, T. Schirmeister, A. Braeuning, D. Lichtenstein, U. A. Hellmich, D. Weikert, M. Heinrich, G. Treccani, M. K. E. Sch fer, G. Nowak, B. N rnberg, C. Alzheimer, C. P. M ller and K. Friedland, Mol. Psychiatry, 2022, 27, 5070-5085.
DOI: 10.1038/s41380-022-01804-3
126Tunable Composition of Mixed Self-Assembled Shell-by-Shell Structures on Nanoparticle Surfaces
A. Eigen, L. M. S. Stiegler, S. Gradl, V. Schneider, V. Wedler, H. Ga , L. M ller, M. Sarcletti, M. R. Heinrich, A. Hirsch, M. Halik, Adv. Mater. Interfaces, 2022, 9, 32, 2201471.
DOI: 10.1002/admi.202201471
125pH-Dependent Conformational Switching of Amide Bonds-from Full trans to Full cis and Vice Versa
R. Thurston, V. Zantop, K. S. Park, H. Maid, A. Seitz, M. R. Heinrich, Org. Lett., 2022, 24, 3488-3492.
DOI: 10.1021/acs.orglett.2c00938
124Current advances in Meerwein-type radical alkene functionalizations
N. Diesendorf, M. R. Heinrich, Synthesis, 2022, 54, 1951 1963.
DOI: 10.1055/s-0040-1719893
123Synthesis of 2-(Chlorodifluoromethyl)indoles for Nucleophilic Halogen Exchange with [18F]Fluoride
L. Bock, S. K. Schulthei , S. Maschauer, R. Lasch, S. Gradl, O. Prante, S. Z. Zard, M. R. Heinrich, Eur. J. Org. Chem., 2021, 46, 6258-6262.
DOI: 10.1002/ejoc.202100937
122Cleavage of organosolv lignin to phenols using nitrogen monoxide and hydrazin
L.-E. Hofmann, L.-M. Altmann, O. Fischer, L. Prusko, G. Xiao, N. Westwood, M. R. Heinrich, ACS Omega, 2021, 6, 30, 19400-19408.
DOI: 10.1021/acsomega.1c00996
121A synthetic route to phenyl diazenes and pyridazinium salts from phenylazosulfonates
S. Gradl, J. K ckenberger, M. Schiller, J. Oppl, M. R. Heinrich, J. Org. Chem 2021, 86, 9, 6228-6238.
DOI: 10.1021/acs.joc.1c00013
1202-Fluoro-5-nitrophenyldiazonium a novel Sanger-type reagent for the versatile functionalization of alcohols
O. Fischer, M. R. Heinrich, Chem. Eur. J. 2021, 27, 5417-5421.
DOI: 10.1002/chem.202100187
119Visible light promoted, catalyst-free radical carbohydroxylation and carboetherification under mild biomimetic condtions
L.-M. Altmann, V. Zantop, P. Wenisch, N. Diesendorf, M. R. Heinrich, Chem. Eur. J. 2021, 27, 2452-2462.
DOI: 10.1002/chem.202004234
118
Shifted selectivity in protonation enables the mild deuteration of arenes through catalytic amounts of Bronsted acids in deuterated methanol
O. Fischer, A. Huber, M. R. Heinrich, J. Org. Chem. 2020, 85, 11856-11866.
DOI: 10.1021acs.joc.0c01604
117Oxidative formation of disulfide bonds by a chemiluminescent 1,2-dioxetane under mild conditions
C. S. Sauer, J. K ckenberger, M. R. Heinrich, J. Org. Chem. 2020, 85, 14, 9331-9338.
DOI: 10.1021/acs.joc.0c00569
116N-Alkylaminoferrocene-Based Prodrugs Targeting Mitochondria of Cancer Cells
V. Reshetnikov, G. H. zkan. S. Daum, C. Janko, C. Alexiou, C. Sauer, M. R. Heinrich, A. Mokhir, Molecules, 2020, 25(11), 2545
DOI: 10.3390/molecules25112545
115Synthesis, biological evaluation and radiosynthesis of buprenorphine-derived phenylazocarboxamides as novel -opioid receptor ligands
J. Kr ll, S. K. Fehler, L. Hofmann, N. Nebel, S. Maschauer, O. Prante, P. Gmeiner, H. Lanig, H. H bner, M. R. Heinrich, ChemMedChem, 2020, 15, 1175.
DOI: 10.1002/cmdc.202000180
114Medication safety in intravenous therapy: A compatibility study and analysis of reaction products of dihydralazine and metamizole
A. K. Koller, O. Fischer, S. Krebs, M. R. Heinrich, F. D rje, Sci. Pharm. 2020, 88(2), 25.
DOI: 10.3390/scipharm88020025
113Regiospecific introduction of halogens on the 2-aminobiphenyl subunit leads to highly potent M3 muscarinic acetylcholine receptor antagonists and weak inverse agonists
O. Fischer, J. Hofmann, H. Rampp, G. Pratsch, A. Bartuschat, J. Kaindl, R. V. Taudte, M. F. Fromm, H. H bner, P. Gmeiner, M. R. Heinrich, J. Med. Chem 2020,
DOI: 10.1021/acs.jmedchem.0c00297
112Sequential cleavage of lignin systems by nitrogen monoxide and hydrazine
L.-E. Hofmann, D. Hofmann, L. Prusko, L.-M. Altmann, M. R. Heinrich, Adv. Synth. Catal. 2020,
DOI: 10.1002/adsc.201901641
111Aryl Radical Selectivity in Biphasic Systems
L.-M. Altmann, M. C. D. F rst, E. I. Gans, V. Zantop, G. Pratsch, M. R. Heinrich, Org. Lett. 2020, 22, 479-482.
DOI: 10.1021/acs.orglett.9b04237
110Benzyl phenylsemicarbazides: a chemistry-driven approach leading to G protein-biased dopamine D4 receptor agonists with high subtype selectivity
A. Pirzer, R. Lasch, H. Friedrich, H. H bner, P. Gmeiner, M. R. Heinrich, J. Med. Chem. 2019, 62 (21), 9658-9679.
DOI: 10.1021/acs.jmedchem.9b01085
109Preparation of fluorophenyl substituted muscarinic receptor ligands with selectivity for M3 over M2.
A. Banerjee, A. Bartuschat, K. Eitel, P. Gmeiner, M. Heinrich, J. Hofmann, H. Huebner, H. Rampp, B. Schaake, B. Kobilka, R. Sunahara, M. J. Clark, I. Fish, B. Shoichet, WO 2019110521, A1 20190613, PCT Int. Appl. 2019.
108Selective functionalization of graphene at defect activated sites by arylazocarboxylic tert-butylesters
C.E. Halbig, R. Lasch, J. Kr ll, A. Pirzer, Z. Wang, J. N. Kirchhof, K. I. Bolotin, M. R. Heinrich, S. Eigler, Angew. Chem. Int. Ed. 2019, 58, 3599-3603.
DOI: 10.1002/anie.201811192
107
Radical carbofluorination of alkenes with arylhydrazines and Selectfluor: Additives, mechanistic pathways and polar effects
A. S. Pirzer, E. M. Alvarez, H. Friedrich, M. R. Heinrich, Chem. Eur. J. 2019, 25, 2786-2792.
DOI: 10.1002/chem.201805256
106Synthesis of Fmoc- and Boc-protected (2S,5S)- and (2R, 5R)-aminomethylprolines
A. Bartuschat, N. Hegmann, M. R. Heinrich, Synthesis, 2019, 51, 976-984.
DOI: 10.1055/s-0037-1610304
105[18]Fluorine-Labeled Pharmaceuticals: Direct Aromatic Fluorination Compared to Multi-Step Strategies (focus review)
J. Kröll, M. R. Heinrich, Asian J. Org. Chem. 2019, 8, 576-590.
DOI: 10.1002/ajoc.201800494
104In situ conformational fixation of the amide bond enables a general access to medium-sized lactams via ring-closing metathesis
N. Hegmann, L. Prusko, N. Diesendorf, M. R. Heinrich, Org. Lett. 2018, 20, 7825-7829.
DOI: 10.1021/acs.orglett.8b03320
103Structure-guided development of selective muscarinic M3 acetylcholine receptor antagonists
H. Liu, J. Hofmann, I. Fish, B. Schaake, K. Eitel, A. Bartuschat, J. Kaindl, H. Rampp, A. Banerjee, H. H bner, M. J. Clark, S. G. Vincent, J. T. Fisher, M. R. Heinrich, K. Hirata, X. Liu, R. K. Sunahara, B. K. Shoichet, B. K. Kobilka, P. Gmeiner, Proc. Natl. Acad. Sci. USA 2018, 115, 12046-12050.
DOI: 10.1073/pnas.1813988115
102Frozen aryldiazonium chlorides in radical reactions with alkenes and arenes
D. Thon, M. C. D. Fürst, L. Altmann, M. R. Heinrich, Tetrahedron 2018, 74, 5289-5294 (Barton Centennial Issue).
DOI: 10.1016/j.tet.2018.05.089
101Molecular mechanisms of biased and probe-dependent signalling at CXCR3 induced by negative allosteric modulators
R. Brox, L. Milanos, N. Saleh, P. Baumeister, A. Buschauer, D. Hofmann, M. R. Heinrich, T. Clark, N. Tschammer, Mol. Pharmacol. 2018, 93, 309-322.
DOI: 10.1124/mol117.110296
100Ullmanns Encyclopedia of Industrial Chemistry: Antiparasitics (P)
M. C. D. Fürst, A. Pirzer, M. R. Heinrich, Wiley-VCH, 2018.
99Nitrogen oxides and nitric acid enable the sustainable hydroxylation and nitrohydroxylation of benzenes under visible light irradiation
L.-E. Hofmann, L. Mach, M. R. Heinrich, J. Org. Chem. 2018, 83, 431-436.
DOI: 10.1021/acs.joc.7b02333
98[18]Fluorophenylazocarboxylates: Design and synthesis of potential radioligands for the dopamine D3 and μ-opioid receptor
N. Nebel, B. Strauch, S. Maschauer, R. Lasch, H. Rampp, S. K. Fehler, L. R. Bock, H. H bner, P. Gmeiner, M. R. Heinrich, O. Prante, ACS Omega 2017, 2, 8649-8659.
DOI: 10.1021/acsomega.7b01374
97Microwave-assisted rapid one-pot synthesis of fused and non-fused indoles and 5-[18F]fluoroindoles from phenylazocarboxylates
J. Kr ll, A. Hubert, N. Nebel, O. Prante,  M. R. Heinrich, Chem. Eur. J. 2017, 23, 16174-16178.
DOI: 10.1002/chem.201703890
96Visible light induced, radical arylations of arenes and heteroarenes with aryldiazonium salts
Michael C. D. F rst, E. Gans, Michael J. B ck,  M. R. Heinrich, Chem. Eur. J. 2017, 23, 15312-15315.
DOI: 10.1002/chem.201703954
95Process for the synthesis of aryldiazonium salts using nitrogen oxides in oxygen-containing gas streams, especially from industrial waste gases
D. Hofmann, J. Hofmann, M. R. Heinrich, EP3173401, WO2017089470.
94Entstickung mit Mehrwert – Stickoxide f r die Herstellung von Farbstoffen und Arzneimitteln
D. Hofmann, M. R. Heinrich, Laborpraxis 2017 (20.06.2017).
93Radical arylation of anilines and pyrroles via aryldiazotates
J. Hofmann, E. Gans, T. Clark, M. R. Heinrich, Chem. Eur. J. 2017, 23, 9647-9656.
DOI: 10.1002/chem.201701429
92Synthesis of spirocyclohexadienones through radical cascade reactions featuring 3-fold carbon-carbon bond formation
N. Hegmann, L. Prusko, M. R. Heinrich, Org. Lett. 2017, 19, 2222-2225, highlighted in Synfacts 07/2017.
DOI: 10.1021/acs.orglett.7b00676
91Strategien zur synthetischen Nutzung von Stickoxiden aus Abgasen
D. Hofmann, M. R. Heinrich, GIT Labor-Fachzeitschrift 2017, Nr. 9, 36.
90Sustainable synthesis of balsalazide and sulfasalazine based on diazotization with low concentrated nitrogen dioxide in air
D. Hofmann, E. Gans, J. Kr ll, M. R. Heinrich, Chem. Eur. J. 2017, 23, 4042-4045 (Hot Paper), highlighted in Synfacts 07/2017.
DOI: 10.1002/chem.201605359
89
Organic chemistry – more radical than ever before
M. R. Heinrich, Tetrahedron 2016, 72, 7655 (preface to the special issue on radical chemistry).
DOI: 10.1016/j.tet.2016.09.064
88Strongly directing substituents in the radical arylation of substituted benzenes
J. Hofmann, T. Clark, M. R. Heinrich, J. Org. Chem. 2016, 81, 9785-9791.
DOI: 10.1021/acs.joc.6b01840
87Recent developments in intramolecular radical arylations of arenes and heteroarenes
J. Hofmann, M. R. Heinrich, Tetrahedron Lett. 2016, 57, 4334-4340 (short review).
DOI:10.1016/j.tetlet.2016.08.034
864-Biphenylalanine- and 3-phenyltyrosine-derived hydroxamid acids as inhibitors of the JumonjiC domain-containing histone demethylase KDM4A
L. Morera, M. Roatsch, M. C. D. F rst, I. Hoffmann, J. Senger,  M. Hau, H. Franz, R. Sch le, M. R. Heinrich, M. Jung,  ChemMedChem 2016, 11, 2063-2083.
DOI: 10.1002/cmdc.201600218
85
Regioselective radical arylation of 3-hydroxypyridines
M. C. D. F rst, L. Bock, M. R. Heinrich, J. Org. Chem. 2016, 81, 5752-5758.
DOI: 10.1021/acs.joc.6b00894
84
Thermally induced carbohydroxylation of styrenes with aryldiazonium salts
S. Kindt, K. Wicht, M. R. Heinrich, Angew. Chem. Int. Ed. 2016, 55, 8744-8747.
DOI: 10.1002/anie.201601656
83
Synthesis of 6-arylpyridin-3-ols via oxidative rearrangement of 5-arylfurfurylamines
M. C. D. F rst, C. S. Sauer, T. Moriyama, A. Kamimura, M. R. Heinrich, Eur. J. Org. Chem. 2016, 3051-3055.
DOI: 10.1002/ejoc.201600377
82Radical arylation of tyrosine residues in peptides
S. K. Fehler, G. Pratsch, C. streicher, M. C. D. F rst, M. Pischetsrieder, M. R. Heinrich, Tetrahedron 2016, 72, 7888-7893.
DOI: 10.1016/j.tet.2016.04.084
81Hydrogen peroxide-promoted Mizoroki-Heck reactions of phenyldiazenes with acrylates, acrylamides and styrenes
R. Lasch, S. K. Fehler, M. R. Heinrich, Org. Lett. 2016, 18, 1586-1589.
DOI: 10.1021/acs.orglett.6b00449
80Recent advances in Meerwein arylation chemistry
S. Kindt, M. R. Heinrich, Synthesis 2016, 48, 1597-1606 (short review).
DOI: 10.1055/s-0035-1561586
79Development of Photoactivatable Allosteric Modulators for the Chemokine Receptor CXCR3
T. H. Admas, V. Bernat, M. R. Heinrich, N. Tschammer, ChemMedChem 2016, 11, 575-584.
DOI: 10.1002/cmdc.201500573
782,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor H1/H4-receptor selectivity
S. G. Hammer, S. Gobleder, F. Naporra, H.-J. Wittmann, S. Elz, M. R. Heinrich, A. Strasser, Bioorg. Med. Chem. Lett. 2016, 26, 292-300.
DOI: 10.1016/j.bmcl.2015.12.035
77Base-induced radical carboamination of non-activated alkenes with aryldiazonium salts
S. Kindt, K. Wicht, M. R. Heinrich, Org. Lett. 2015, 17, 6122-6125.
DOI: 10.1021/acs.orglett.5b03143
76Denitrification combined with diazotization of anilines and the synthesis of 4 chlorobiphenyl-2,5-diamine and 1-chloro-4-iodobenzene
D. Hofmann, J. Hofmann, L. Hofmann, L. E. Hofmann, M. R. Heinrich, Org. Process Res. Dev. 2015, 19, 2075-2084.
DOI: 10.1021/acs.oprd.5b00298
75Schnelle und effiziente Herstellung vielseitig einsetzbarer 18F-markierter Vorl ufer für die Synthese radiomarkierter Verbindungen
S. K. Fehler, S. Maschauer, O. Prante, M. R. Heinrich, DE102014017352A1.
74Zinc-mediated allylation and benzylation of phenylazocarboxylic esters
R. Lasch, M. R. Heinrich, J. Org. Chem. 2015, 80, 10412-10420.
DOI: 10.1021/acs.joc.5b01978
73Oxidative nitration of styrenes for the recycling of low-concentrated nitrogen dioxide in air
D. Hofmann, C. de Salas,  M. R. Heinrich, ChemSusChem 2015, 8, 3167-3175.
DOI: 10.1002/cssc.201500188
72Switching and conformational fixation of amides through proximate positive charges
A. L. Bartuschat, K. Wicht, M. R. Heinrich, Angew. Chem. Int. Ed. 2015, 54, 10294 10298.
DOI: 10.1002/ange.201502474; DOI: 10.1002/anie.201502474
71Cycloadditions to phenylazocarboxylic esters: a new access to highly substituted triazoles
R. Lasch, M. R. Heinrich, Tetrahedron 2015, 71, 4282-4295.
DOI: 10.1016/j.tet.2015.04.078
70Ligand biased and probe-dependend modulation of the chemokine receptor CXCR3 signaling by negative allosteric modulators
V. Bernat, R. Brox, M. R. Heinrich, Y. Auberson, N. Tschammer, ChemMedChem 2015, 10, 556-574.
DOI: 10.1002/cmdc.201402507
69Fluoro-substituted phenylazocarboxamides: dopaminergic behavior and N-arylating properties for irreversible binding
A. L. Bartuschat, T. Schellhorn, H. H bner, P. Gmeiner, M. R. Heinrich, Bioorg. Med. Chem. 2015, 23, 3938-3947.
DOI: 10.1016/j.bmc.2014.12.012
68From a natural product to aryl radical chemistry
S. K. Fehler, M. R. Heinrich, Synlett 2015, 580-603 (account article).
DOI: 10.1055/s-0034-1378945
67Synthesis of dibenzo[c,e][1,2]diazocines – a new group of eight-membered cyclic azo compounds
T. Nokubi, S. Kindt, T. Clark, A. Kamimura, M. R. Heinrich, Tetrahedron Lett. 2015, 56, 316-320.
DOI: 10.1016/j.tetlet.2014.11.064
66Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues as potential dopamine D3 receptor PET ligands
N. Nebel, S. Maschauer, A. L. Bartuschat, S. K. Fehler, H. H bner, P. Gmeiner, T. Kuwert, M. R. Heinrich, O. Prante, C. Hocke, Bioorg. Med. Chem. Lett. 2014, 24, 5399-5403.
DOI: 10.1016/j.bmcl.2014.10.043
65Intermolecular radical carbofluorination of non-activated alkenes
S. Kindt, M. R. Heinrich, Chem. Eur. J. 2014, 20, 15344-15348.
DOI: 10.1002/chem.201405229
64Synthesis of 7-arylquinolinones and 6-arylindoles from 3-aminobiphenyls through regioselective cyclization reactions
S. G. Hammer, M. R. Heinrich, Tetrahedron 2014, 70, 8114-8121.
DOI: 10.1016/j.tet.2014.08.012
63The trapping of phenyldiazenes in cycloaddition reactions
S. K. Fehler, G. Pratsch, M. R. Heinrich, Angew. Chem. 2014, 126, 11543 11548, Angew. Chem. Int. Ed. 2014, 53, 11361-11365.
DOI: 10.1002/ange.201406175; DOI: 10.1002/anie.201406175
62Fixation and recycling of nitrogen monoxide through carbonitrosation reactions
C. de Salas, M. R. Heinrich, Green Chem. 2014, 16, 2982-2987.
DOI: 10.1039/C3GC42432D
61Manganese(IV)-mediated hydroperoxyarylation of alkenes with arylhydrazines and dioxygen from air
S. Kindt, H. Jasch, M. R. Heinrich, Chem. Eur. J. 2014, 20, 6251 6255.
DOI: 10.1002/chem.201400064
60Radiosynthesis and validation of 18F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain
P. Cumming, S. Maschauer, P. Riss, N. Tschammer, S. Fehler, M. R. Heinrich, T. Kuwert, O. Prante, J. Cereb. Blood Flow Metab. 2014, 34, 1148-1156.
DOI: 10.1038/jcbfm.2014.63
59Oxidative radical arylation of anilines with arylhydrazines and dioxygen from air
J. Hofmann, H. Jasch, M. R. Heinrich, J. Org. Chem. 2014, 79, 2314 2320.
DOI: 10.1021/jo500063r
58Alanine-glyoxylate aminotransferase 2 (AGXT2) polymorphisms have considerable impact on methylarginine and beta-aminoisobutyrate metabolism in healthy volunteers
A. Kittel, F. M ller, J. K nig, M. Mieth, S. Bode-B ger, A. Kralj, M. R. Heinrich, M. F. Fromm, R. Maas, PLOS ONE 2014, 9, e88544.
DOI: 10.1371/journal.pone.0088544
57Synthesis and biological evaluation of biphenyl amides that modulate the US28 receptor
A. Kralj, E. Kurt, N. Tschammer, M. R. Heinrich, ChemMedChem 2014, 9, 151-168.
DOI: 10.1002/cmdc.201300369
56Fast and efficient 18F-labeling via [18F]fluorophenylazocarboxylic esters
S. Fehler, S. Maschauer, S. H fling, A. Bartuschat, N. Tschammmer, H. H bner, P. Gmeiner, O. Prante, M. R. Heinrich, Chem. Eur. J. 2014, 20, 370-375.
DOI: 10.1002/chem.201303409
55Carbon-carbon bond forming reactions involving aryl radicals
S. Hammer, M. R. Heinrich, Comprehensive Organic Synthesis, 2014
ISBN-10: 0-080-97742-1; ISBN-13: 978-0-080-97742-3.
54Method for synthesising aminobiphenyls using aryl hydrazines
M. Heinrich, H. Jasch, S. H fling, WO2013132006.
53Studies on the synthesis and biosynthesis of the fungal alkaloid necatorone
J. Carstens, M. R. Heinrich, W. Steglich, Tetrahedron Lett. 2013, 54, 5445-5447.
DOI: 10.1016/j.tetlet.2013.07.118
52Enzymatic kinetic resolution and racemization of 2-(tetramethylpiperidine-1-oxyl)ethanols
A. Prechter, M. R. Heinrich, Eur. J. Org. Chem. 2013, 5585-5589.
DOI: 10.1002/ejoc.201300661
51Development of flavonoid-based inverse agonists of the key signaling receptor US28 of Human Cytomegalovirus
A. Kralj, M.-T. Nguyen, N. Tschammer, N. Ocampo, Q. Gesiotto, M. R. Heinrich, O. Phanstiel,  J. Med. Chem. 2013, 56, 5019-5032.
DOI: 10.1021/jm4003457
50Twofold carbon-carbon bond formation via intramolecular and intermolecular radical reactions of aryl diazonium salts
H. Jasch, Y. Landais, M. R. Heinrich, Chem. Eur. J. 2013, 19, 8411-8416.
DOI: 10.1002/chem.201300354
49Process for the synthesis of aminobiphenylene
M. Heinrich, G. Pratsch, WO2012120003.
48Verfahren zur Synthese von Aryloximen unter Verwendung von Stickstoffmonoxid
M. Heinrich, C. de Salas, DE102012010413.
47Regioselective radical arylation of anilines with arylhydrazines
H. Jasch, J. Scheumann, M. R. Heinrich, J. Org. Chem. 2012, 77, 10699-10706.
DOI: 10.1021/jo301980j
46Synthesis and Application of the First Radioligand Targeting the Allosteric Binding Pocket of Chemokine Receptor CXCR3
V. Bernat, M. R. Heinrich, P. Baumeister, A. Buschauer, N. Tschammer, ChemMedChem 2012, 7, 1481-1489.
DOI: 10.1002/cmdc.201200184
45The Gomberg-Bachmann Reaction for the Arylation of Anilines with Aryl Diazotates
G. Pratsch, T. Wallaschkowski, M. R. Heinrich, Chem. Eur. J. 2012, 18. 11555-11559.
DOI: 10.1002/chem.201200430
44Synthesis of (S)-(+)-cericlamine through lipase-catalyzed aminolysis of azo acetates
A. Prechter, H. Gr ger, M. R. Heinrich, Org. Biomol. Chem. 2012, 10, 3384-3387.
DOI: 10.1039/C2OB25247C
43Synthesis and biological evaluation of 3-aryltyramines as fragments binding to BACE-1 and BACE-2
S. K. Fehler, G. Pratsch, W. Huber, A. Gast, R. Hochstrasser, M. Hennig, M. R. Heinrich, Tetrahedron Lett. 2012, 53, 2189-2194.
DOI: 10.1016/j.tetlet.2012.02.070
42Nucleophilic substitutions and radical reactions of phenylazocarboxylates
H. Jasch, S. B. H fling, M. R. Heinrich, J. Org. Chem. 2012, 77, 1520-1532.
DOI: 10.1021/jo202406k
41Modern developments in aryl radical chemistry
G. Pratsch, M. R. Heinrich, Topics in Current Chemistry 2012, 320 (Eds. M. R. Heinrich, A. Gans uer), 33-60.
DOI: 10.1007/128_2011_127
40Tin Hydrides and Functional Group Transformations
H. Jasch, M. R. Heinrich, Encyclopedia of Radicals in Chemistry, Biology and Materials, Eds. C. Chatgilialoglu, A. Studer, 1st ed., John Wiley & Sons, 2012.
ISBN-10: 0-470-97125-8; ISBN-13: 978-0-470-97125-3
39Verfahren zur Herstellung von enantiomerenangereicherten Azoverbindungen, Aminoalkoholen und Aminos uren mit einem quart ren Kohlenstoffzentrum
F. Dietz, H. Gr ger, M. Heinrich, A. Prechter, DE102011101183.
38Identification of novel allosteric modulators for the G-protein coupled US28 receptor of human cytomegalovirus
A. Kralj, A. Wetzel, S. Mahmoudian, T. Stamminger, N. Tschammer, M. R. Heinrich, Bioorg. Med. Chem. Lett. 2011, 21, 5446-5450.
DOI: 10.1016/j.bmcl.2011.06.120
37Radical carbonitrosation and recycling of the waste gas nitrogen monoxide
C. de Salas, O. Blank, M. R. Heinrich, Chem. Eur. J. 2011, 17, 9306-9310.
DOI: 10.1002/chem.201101565
36Hydrogen peroxide and arenediazonium salts as reagents for a radical Beckmann-type rearrangement
A. Prechter, M. R. Heinrich, Synthesis 2011, 10, 1515-1525.
DOI: 10.1055/s-0030-1260006
35Radical arylation of tyrosine and its application in the synthesis of a highly selective neurotensin receptor 2 ligand
G. Pratsch, J. F. Unfried, J. Einsiedel, M. Plomer, H. H bner, P. Gmeiner, M. R. Heinrich, Org. Biomol. Chem. 2011, 9, 3746-3752.
DOI: 10.1039/c1ob05292f
34Hydroxy- and aminophenyl radicals from arenediazonium salts
G. Pratsch, C. A. Anger, K. Ritter, M. R. Heinrich, Chem. Eur. J. 2011. 17, 4104-4108.
DOI: 10.1002/chem.201003713
33Nitrogen-centered radical scavengers
S. B. H fling, M. R. Heinrich, Synthesis 2011, 173-189.
DOI: 10.1055/s-0030-1258305
32Chiral azo compounds: Enantioselective analysis and transformations into β-amino alcohols and α-amino acidswith a quaternary stereocenter
F. R. Dietz, A. Prechter, H. Gr ger, M. R. Heinrich, Tetrahedron Lett. 2010, 52, 655-657.
DOI: 10.1016/j.tetlet.2010.11.137
31Method for arylation ring-substituted phenols and phenylethers
M. Heinrich, A. Wetzel, WO2010112211.
30Method for producing 3-aminobiphenylene
M. Heinrich, A. Wetzel, WO2010037531.
29Method for producing aminobiphenylene
M. Heinrich, A. Wetzel, M. Keil, M. Rack, T. Ziercke, WO201000856.
28Synthesis, biological evaluation and radiolabeling by 18F-fluoroarylation of a dopamine D3 selective ligand as prospective imaging probe for PET
S. B. H fling, S. Maschauer, H. H bner, P. Gmeiner, H.-J. Wester, O. Prante, M. R. Heinrich, Bioorg. Med. Chem. Lett. 2010, 20, 6933-6937.
DOI: 10.1016/j.bmcl.2010.09.142
274-Substituted tert-butyl phenylazocarboxylates – synthetic equivalents for the para-phenyl radical cation
S. B. H fling, A. L. Bartuschat, M. R. Heinrich, Angew. Chem. 2010, 122, 9963-9966, Angew. Chem. Int. Ed. 2010, 49, 9769-9772.
DOI: 10.1002/ange.201004508; DOI: 10.1002/anie.201004508
26Radical arylation of phenols, phenyl ethers, and furans
A. Wetzel, G. Pratsch, R. Kolb, M. R. Heinrich, Chem. Eur. J. 2010, 16, 2547-2556.
DOI: 10.1002/chem.200902927
25Hydroperoxides and aryl diazonium salts as reagents for the functionalization of non-activated olefins
O. Blank, N. Raschke, M. R. Heinrich, Tetrahedron Lett. 2010, 51, 1758-1760.
DOI: 10.1016/j.tetlet.2010.01.098
24Intermolecular olefin functionalizations involving aryl radicals generated from arenediazonium salts
M. R. Heinrich, Chem. Eur. J. 2009, 15, 820-833.
DOI: 10.1002/chem.200801306
23Synthesis of amino- and hydroxybiphenyls by a radical chain reaction of arenediazonium salts
A. Wetzel, V. Ehrhardt, M. R. Heinrich, Angew. Chem. 2008, 120, 9270-9273, Angew. Chem. Int. Ed. 2008, 47, 9130-9133.
DOI: 10.1002/ange.200803785; DOI: 10.1002/anie.200803785
22Radiochemical [18F]fluoroarylation of unsaturated α-, β- and γ-amino acids, application to a radiolabeledderivate of baclofen
S. B. H fling, C. Hultsch, H.-J. Wester, M. R. Heinrich, Tetrahedron 2008, 64, 11846-11851.
DOI: 10.1016/j.tet.2008.07.117
21Radical carbodiazenylation a convenient and effective method to achieve carboamination of non-activated olefins
O. Blank, A. Wetzel, D. Ullrich, M. R. Heinrich, Eur. J. Org. Chem. 2008, 3179-3189.
DOI: 10.1002/ejoc.200800250
20Radical fluoroarylation in radiochemical synthesis
 C. Hultsch, O. Blank, H.-J. Wester, M. R. Heinrich, Tetrahedron Lett. 2008, 49, 1881-1883.
DOI: 10.1016/j.tetlet.2007.12.128
19Allylation and vinylation of aryl radicals generated from diazonium salts
M. R. Heinrich, O. Blank, D. Ullrich, M. Kirschstein, J. Org. Chem. 2007, 72, 9609-9616.
DOI: 10.1021/jo701717k
18Intermolecular radical carboaminohydroxylation of olefins with aryl diazonium salts and TEMPO
M. R. Heinrich, A. Wetzel, M. Kirschstein, Org. Lett. 2007, 9, 3833-3835, Synfacts 2007, 1303.
DOI: 10.1021/ol701622d
17Synthesis of 2-fluorotetralones by oxidative radical cyclization of α-fluoroacetophenones and olefins
 M. R. Heinrich, Tetrahedron Lett. 2007, 48, 3895-3900.
DOI: 10.1016/j.tetlet.2007.03.128
16Oxidative and reductive carbodiazenylation of nonactivated olefins
M. R. Heinrich, O. Blank, A. Wetzel, J. Org. Chem. 2007, 72, 476-484.
DOI: 10.1021/jo061919p
15A new approach to the stereoselective carbodiazenylation of olefins by macrocyclization
M. R. Heinrich, O. Blank, A. Wetzel, Synlett 2006, 3352-3354.
DOI: 10.1055/s-2006-951556
14Carbodiazenylation of olefins by radical iodine transfer and addition to arenediazonium salts
 O. Blank, M. R. Heinrich, Eur. J. Org. Chem. 2006, 4331-4334.
DOI: 10.1002/ejoc.200600528
13Reductive carbodiazenylation of nonactivated olefins via aryl diazonium salts
M. R. Heinrich, O. Blank, S. W lfel, Org. Lett. 2006, 8, 3323-3325, Synfacts 2006, 1045.
DOI: 10.1021/ol0611393
12Photochemical generation and trapping of radicals from bisphenyl carbodiazone
M. R. Heinrich, M. Kirschstein, Tetrahedron Lett. 2006, 47, 2115-2118.
DOI: 10.1016/j.tetlet.2006.01.128
11Generation and ring opening of aziridine N-carbonyl radicals
M. R. Heinrich, I. P rez-Mart n, S. Z. Zard, Chem. Commun. 2005, 5928-5930.
DOI: 10.1039/b512956g
10A convergent approach to γ-carbonyl vinyl boronates
 M. R. Heinrich, L. A. Sharp, S. Z. Zard, Chem. Commun. 2005, 3077-3079.
DOI: 10.1039/b502885j
9Generation and intermolecular capture of cyclopropylacyl radicals
M. R. Heinrich, S. Z. Zard, Org. Lett. 2004, 6, 4969-4972.
DOI: 10.1021/ol047892i
8Enhancing the catalytic activity of 4-(dialkylamino)pyridines by conformational fixation
 M. R. Heinrich, H. S. Klisa, H. Mayr, W. Steglich, H. Zipse, Angew. Chem. 2003, 115, 4975-4977, Angew. Chem. Int. Ed. 2003, 42, 4826-4828.
DOI: 10.1002/ange.200352289; DOI: 10.1002/anie.200352289
7Total synthesis of the marine alkaloid halitulin
M. R. Heinrich, W. Steglich, M. G. Banwell, Y. Kashman, Tetrahedron 2003, 59, 9239-9247.
DOI: 10.1016/j.tet.2003.02.005
6Effective syntheses of quinoline-7,8-diol, 5-amino-L-DOPA, and 3-(7,8-dihydroxyquinolin-5-yl)-L-alanine
M. R. Heinrich, W. Steglich, Tetrahedron 2003, 59, 9231-9237.
DOI: 10.1016/j.tet.2003.02.004
5Revision of the structure of haliclorensin to (S)-7-methyl-1,5-diazacyclotetradecane and confirmation of the new structure by synthesis
 M. R. Heinrich, Y. Kashman, P. Spiteller, W. Steglich, Tetrahedron 2001, 57, 9973-9978.
DOI: 10.1016/S0040-4020(01)01020-1
4Synthesis of (-)-(3S)-1-(3-aminopropyl)-3-methylazacyclo-decane, the structure proposed for the marine alkaloid haliclorensin
M. R. Heinrich, W. Steglich, Tetrahedron Lett. 2001, 42, 3287-3289.
DOI: 10.1016/S0040-4039(01)00435-X
3Novel approach to the chemical bath deposition of chalcogenide semiconductors
 D. S. Boyle, A. Bayer, M. R. Heinrich, O. Robbe, P. O Brien, Thin Solid Films 2000, 361/362, 150-154.
DOI: 10.1016/S0040-6090(99)00789-0
2Developing environmentally benign routes for semiconductor synthesis: improved approaches to  thesolution deposition of cadmium sulfide for solar cell applications
A. Bayer, D. S. Boyle, M. R. Heinrich, D. J. Otway, O. Robbe, P. O Brien, Green Chemistry 2000, 2, 79-86.
DOI: 10.1039/A909257I
1A novel method for the synthesis of the ternary thin film semiconductor cadmium zinc sulfide from acidic chemical baths
D. S. Boyle, O. Robbe, D. P. Halliday, M. R. Heinrich, A. Bayer, P. O Brien, D. J. Otway, M. D. G. Potter, Journal of Materials Chemistry 2000, 10, 2439-2441.
DOI: 10.1039/B005544L

7